41 results
Warfarin and DOAC Pharmacology
Warfarin - Dabigatran - Rivaroxaban - Apixaban - Edoxaban
Target - Prodrug - Bioavailability
Pharmacology Warfarin - Dabigatran ... Rivaroxaban - Apixaban - Edoxaban ... comparison #table #dabigatran ... rivaroxaban #apixaban #edoxaban
DOAC Cheat Sheet
 • Apixaban, Dabigatran, Edoxaban, Rivaroxaban
 • Renal Dosing
 • Common Drug interactions
 •
Sheet • Apixaban, Dabigatran ... , Edoxaban, Rivaroxaban
Oral anticoagulant dosing and bridging for VTE

- Dr. Joseph Shatzel @Clotmaster 

#VTE #DOAC #Bridging #Dosing #Oral
Anticoagulation #Dabigatran ... #Rivaroxaban #Edoxaban
Switching Between Anticoagulants and DOACs
VKA, Dabigatran, Rivaroxaban, Apixaban, Edoxaban, Betrixaban, DOAC, Parenteral anticoagulant

DOI: 10.1161/JAHA.120.017559

#Anticoagulants #DOACs #anticoagulation
and DOACs VKA, Dabigatran ... Rivaroxaban, Apixaban, Edoxaban
DOAC: Cheat Sheet - Atrial Fibrillation, VTE Prophylaxis, VTE and Renal Dosing

Renal Dosing:
Apixaban (25% renal clearance):
patients 5mg bid Dabigatran ... if CrCl < 50) Edoxaban ... #Rivaroxaban #Dabigatran ... #Edoxaban #NOAC
Anticoagulants Common Reversal Agents
 - Warfarin (Coumadin) → Vitamin K (Phytonadione), 4-factor PCC (Kcentra)
 - Heparin/LMWH
Protamine sulfate - Dabigatran ... Betrixaban (Bevyxxa), Edoxaban
Pharmacokinetic Characteristics and Primary Routes of Clearance of Oral Anticoagulant Agents

Warfarin - 100% Hepatic, 0% Renal
Apixaban
Hepatic, 25% Renal Dabigatran ... Hepatic, 80% Renal Edoxaban
Coagulation Cascade - Actions of Anticoagulants
 • Heparin: Unfractionated heparin, Enoxaparin, Daltaparin
 • Fondaparinux
 • Direct
Rivaroxaban, Apixaban, Edoxaban ... Inhibitors: Argatroban, Dabigatran
Effect of Anticoagulants on Coagulation Tests
PT / INR, aPTT, Anti-Xa Activity, Activated Clotting Time, Thrombin Time,
Rivaroxaban Apixaban, Edoxaban ... Argatroban Dabigatran
Anticoagulant Sites of Absorption
Apixaban - Primarily proximal small intestine; some gastric absorption
Dabigatran - Lower stomach and
gastric absorption Dabigatran ... and duodenum Edoxaban