Muscarinic Receptor Agonists and Antagonists 
Muscarinic Receptor Agonists
Methacholine
 • Diagnosis of bronchial airway
Carbachol
 • Glaucorna (topical administration)
Bethanechol
 • Ileus (postoperative, neurogenic)
 • Urinary retention
Pilocarpine
 • Glaucorna (topical administration)
 • Xerostomia due to Sjögren syndrome, Head and neck irradiation
Cevimeline
 • Xerostomia due to Sjögren syndrome
Muscarinic Receptor Antagonists
Atropine
 • Acute symptomatic bradycardia (e.g., AV block)
 • Cholinesterase inhibitor intoxication
 • Aspiration prophylaxis
Scopolamine
 • Motion sickness
Homatropine, cyclopentolate, tropicamide
 • Ophthalmological examination (cycloplegia and mydriasis induction)
Ipratropium, tiotropium, aclidinium. umeclidinium
 • COPD
 • Rhinorrhea (ipratropium)
Pirenzepine, telenzepine
 • Peptic ulcer disease (notin US.)
Oxybutynin, trospium, darifenacin, solifenacin, tolterodine, fesoterodine
 • Overactive bladder, enuresis, neurogenic bladder
Glycopyrrolate
 • Duodenal ulcer
 • Sialorrhea
Dicyclomine, hyoscyamine
 • Diarrhea-predominant irritable bowel syndrome (IBS)
Trihexyphenidyl, benztropine
 • Parkinson disease

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