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Lamotrigine Pharmacokinetics and Drug-Drug Interactions

- Drs. Ashley & Brooke Barlow @theABofPharmaC

#Lamotrigine #Pharmacokinetics #DrugDrug #Interactions #Pharmacology #SideEffects
Lamotrigine Pharmacokinetics ... theABofPharmaC #Lamotrigine ... #SideEffects #Lamictal
Pharmacology of Antipsychotic Drugs for Bipolar Disorder
 • PHENOTHIAZINES: Chlorpromazine, Fluphenazine, Thioridazine
 • THIOXANTHENE: Thiothixene
 •
Carbamazepine, Lamotrigine
Trigeminal Neuralgia [Tic douloureux] 
Clinical 
 • Excruciating paroxysmal pain 
 • Right > Left side
• Gabapentin, Lamotrigine
Antiseizure Drugs 
Sodium Channel Blockers: Carbamazepine, Oxcarbazepine, Eslicarbazepine, Lamotrigine, Lacosamide, Phenytoin, fosphenytoin
Broad Spectrum: Valproate, Levetiracetam, Brivaracetam,
Eslicarbazepine, Lamotrigine
Stevens Johnson Syndrome and Toxic Epidermal Necrolysis - Causative Medications 
and Level of Suspicion 

High Risk:
Antigout:
carbamazepine, lamotrigine
Intravenous Lipid Emulsion (ILE) Therapy

ILE is a treatment for severe toxicity from local anesthetics. In addition,
anticonvulsants (lamotrigine
Anticonvulsants as Mood Stabilizers: Mechanism and Side-effect
Examples: Valproate, Carbamazepine, Lamotrigine
 • Mild anticholinergic effect -> Drowsiness
Carbamazepine, Lamotrigine
Anti-Seizure Medication Guide - Common Uses and Side Effects

acetazolamide 
brivaracetam 
carbamazepine 
clobazam 
clonazepam 
clorazepate 
corticotropin injection
diazepam
lacosamide lamotrigine
Causes of Fever: IMADE Mnemonic
INFECTION
 • Infection 1.0 - Common & Localizing: Base Rate
 • Infection
DRUGS • SJS-TEN: lamotrigine ... carbamezapine. lamotrigine
Drugs Related to DRESS Syndrome / DIHS 

The cases that were more consistent with DRESS/DIHS were
zonisamide and lamotrigine